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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T20712 | Conessine | Conessinum,Wrightine,Roquessine,Neriine,Konessin | Histamine Receptor |
Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity. | |||
T6164 | Ciproxifan | FUB-359 | Histamine Receptor |
Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM). | |||
T41247 | Thioperamide maleate | MR-12842 maleate | Histamine Receptor |
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31 nM). | |||
T22864 | Immethridine dihydrobromide | Others | |
Immethridine dihydrobromide is a histamine H3 receptor agonist. | |||
T10499 | H3 receptor-MO-1 | Histamine Receptor | |
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders. | |||
T27678 | JNJ-39220675 | JNJ39220675 | |
JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats. | |||
T67828 | Enerisant | ||
Enerisant is an antagonist/inverse agonist of histamine H3 receptor.In vitro studies have shown that enerisant is a potent, highly selective, and competitive antagonist for the histamine H3 receptor, with a more than 3,0... | |||
T79500L | KSK94 FA | KSK94 FA(2566716-07-0 Free base) | Histamine Receptor |
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity. | |||
TQ0066 | GSK189254A | GSK189254 | Histamine Receptor |
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3). | |||
T7413 | JNJ-5207852 | Histamine Receptor | |
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. | |||
T8822 | JNJ-5207852 dihydrochloride | Histamine Receptor | |
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. | |||
T7176 | Pitolisant hydrochloride | BF 2649,Ciproxidine | Histamine Receptor |
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM). | |||
T77593 | KSK67 | Sigma receptor | |
KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki values of 3.2, 1531, and 101 nM, respectively.KSK67 can be used ... | |||
T61213 | PF-03654764 | Histamine Receptor | |
PF-03654764 is an orally active, potent, and selective histamine H3 receptor antagonist that inhibits human H3 and rat H3 with Ki values of 1.2 nM and 7.9 nM, respectively.PF-03654764 is often co-administered with Fexofe... | |||
T70489 | Enerisant HCl | P450 , Histamine Receptor | |
Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins. | |||
T79499 | KSK68 | Histamine Receptor | |
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 receptors.KSK68 can be used in the study of pain related diseases... | |||
T12054L | MK-0249 FA | MK-0249 FA(862309-06-6 Free base) | Histamine Receptor |
MK-0249 FA is an orally active, selective and potent histamine H3 inverse agonist for the study of attention deficit, hyperactivity disorder neurodivergent and cognitive disorders in adults. | |||
T14087 | ABT-239 | TRP/TRPV Channel | |
ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists. It also acts as a transient receptor potential vanilloid type 1 (TRPV1) antagonist. | |||
T32191 | Irdabisant | CEP-26401,CEP 26401,CEP26401 | Histamine Receptor |
Irdabisant (CEP-26401) (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R Ki= 7.2 nM, human H3R Ki= 2.0 nM). Irdabisant ex... | |||
T0246 | Betahistine dihydrochloride | PT-9,Betahistine 2HCl | Histamine Receptor |
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator. |