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Search Results for " histamine h3 "

20

Compounds

Cat No. Product Name Synonyms Targets
T20712 Conessine Conessinum,Wrightine,Roquessine,Neriine,Konessin Histamine Receptor
Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
T6164 Ciproxifan FUB-359 Histamine Receptor
Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
T41247 Thioperamide maleate MR-12842 maleate Histamine Receptor
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31 nM).
T22864 Immethridine dihydrobromide Others
Immethridine dihydrobromide is a histamine H3 receptor agonist.
T10499 H3 receptor-MO-1 Histamine Receptor
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
T27678 JNJ-39220675 JNJ39220675
JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.
T67828 Enerisant
Enerisant is an antagonist/inverse agonist of histamine H3 receptor.In vitro studies have shown that enerisant is a potent, highly selective, and competitive antagonist for the histamine H3 receptor, with a more than 3,0...
T79500L KSK94 FA KSK94 FA(2566716-07-0 Free base) Histamine Receptor
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.
TQ0066 GSK189254A GSK189254 Histamine Receptor
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
T7413 JNJ-5207852 Histamine Receptor
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T8822 JNJ-5207852 dihydrochloride Histamine Receptor
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T7176 Pitolisant hydrochloride BF 2649,Ciproxidine Histamine Receptor
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
T77593 KSK67 Sigma receptor
KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki values of 3.2, 1531, and 101 nM, respectively.KSK67 can be used ...
T61213 PF-03654764 Histamine Receptor
PF-03654764 is an orally active, potent, and selective histamine H3 receptor antagonist that inhibits human H3 and rat H3 with Ki values of 1.2 nM and 7.9 nM, respectively.PF-03654764 is often co-administered with Fexofe...
T70489 Enerisant HCl P450 , Histamine Receptor
Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins.
T79499 KSK68 Histamine Receptor
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 receptors.KSK68 can be used in the study of pain related diseases...
T12054L MK-0249 FA MK-0249 FA(862309-06-6 Free base) Histamine Receptor
MK-0249 FA is an orally active, selective and potent histamine H3 inverse agonist for the study of attention deficit, hyperactivity disorder neurodivergent and cognitive disorders in adults.
T14087 ABT-239 TRP/TRPV Channel
ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists. It also acts as a transient receptor potential vanilloid type 1 (TRPV1) antagonist.
T32191 Irdabisant CEP-26401,CEP 26401,CEP26401 Histamine Receptor
Irdabisant (CEP-26401) (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R Ki= 7.2 nM, human H3R Ki= 2.0 nM). Irdabisant ex...
T0246 Betahistine dihydrochloride PT-9,Betahistine 2HCl Histamine Receptor
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.
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